Desmethylmoramide

Opioid analgesic drug

Desmethylmoramide
Names

Preferred IUPAC name 4-(Morpholin-4-yl)-2,2-diphenyl-1-(pyrrolidin-1-yl)butan-1-one
Identifiers
CAS Number	1767-88-0^Y
3D model (JSmol)	Interactive image
ChEMBL	ChEMBL2106152
ChemSpider	178501
PubChem CID	206005
UNII	9B1Z1V29C3^Y
CompTox Dashboard (EPA)	DTXSID60170172
InChI InChI=1S/C24H30N2O2/c27-23(26-14-7-8-15-26)24(21-9-3-1-4-10-21,22-11-5-2-6-12-22)13-16-25-17-19-28-20-18-25/h1-6,9-12H,7-8,13-20H2 Key: JRPANCYSRUEJDY-UHFFFAOYSA-N
SMILES C1CCN(C1)C(=O)C(CCN2CCOCC2)(C3=CC=CC=C3)C4=CC=CC=C4
Properties
Chemical formula	C₂₄H₃₀N₂O₂
Molar mass	378.516 g·mol⁻¹
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa). Infobox references

Chemical compound

Desmethylmoramide (INN) is an opioid analgesic related to dextromoramide (the active (+)-isomer of moramide) that was synthesized and characterized in the late 1950s but was never marketed.^[1]^[2]^[3]

References

^ Elks J (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. pp. 363–. ISBN 978-1-4757-2085-3.
^ Morton IK, Hall JM (6 December 2012). Concise Dictionary of Pharmacological Agents: Properties and Synonyms. Springer Science & Business Media. pp. 94–. ISBN 978-94-011-4439-1.
^ Janssen PA, Jageneau AH (June 1957). "A new series of potent analgesics: dextro 2:2-diphenyl-3-methyl-4-morpholino-butyrylpyrrolidine and related amides. I. Chemical structure and pharmacological activity". The Journal of Pharmacy and Pharmacology. 9 (6): 381–400. doi:10.1111/j.2042-7158.1957.tb12290.x. PMID 13439527. S2CID 58956931.